Structure-Activity Relationship Study of Nonpeptideδ-Opioid Receptor Ligands

Activity Relationship ◽

Receptor Ligands ◽

Structure Activity ◽

Opioid Receptor Ligands ◽

Structure activity relationship studies of 17-cyclopropylmethyl-3,14β-dihydroxy-4,5α-epoxy-6α-(isoquinoline-3′-carboxamido)morphinan (NAQ) analogues as potent opioid receptor ligands: Preliminary results on the role of electronic characteristics for affinity and function

Bioorganic & Medicinal Chemistry Letters ◽

10.1016/j.bmcl.2013.07.043 ◽

2013 ◽

Vol 23 (18) ◽

pp. 5045-5048 ◽

Cited By ~ 7

Author(s):

Yunyun Yuan ◽

Orgil Elbegdorj ◽

Irina O. Beletskaya ◽

Dana E. Selley ◽

Yan Zhang

Keyword(s):

Opioid Receptor ◽

Activity Relationship ◽

Receptor Ligands ◽

Preliminary Results ◽

Structure Activity ◽

Opioid Receptor Ligands ◽

And Function

Structure-activity Relationship, Conformation and Pharmacology Studies of Morphiceptin Analogues - Selective μ-Opioid Receptor Ligands

Mini-Reviews in Medicinal Chemistry ◽

10.2174/1389557023405567 ◽

2002 ◽

Vol 2 (6) ◽

pp. 565-572 ◽

Cited By ~ 11

Author(s):

Anna Janecka ◽

Jakub Fichna ◽

Marek Mirowski ◽

Tomasz Janecki

Keyword(s):

Opioid Receptor ◽

Activity Relationship ◽

Receptor Ligands ◽

Structure Activity ◽

Opioid Receptor Ligands

A Structure–Activity Relationship Study and Combinatorial Synthetic Approach of C-Terminal Modified Bifunctional Peptides That Are δ/μ Opioid Receptor Agonists and Neurokinin 1 Receptor Antagonists

Journal of Medicinal Chemistry ◽

10.1021/jm070332f ◽

2008 ◽

Vol 51 (5) ◽

pp. 1369-1376 ◽

Cited By ~ 36

Author(s):

Takashi Yamamoto ◽

Padma Nair ◽

Josef Vagner ◽

Tally Largent-Milnes ◽

Peg Davis ◽

...

Keyword(s):

Opioid Receptor ◽

Activity Relationship ◽

Synthetic Approach ◽

Neurokinin 1 Receptor ◽

Structure Activity ◽

Μ Opioid Receptor ◽

Relationship Study ◽

Neurokinin 1 ◽

Opioid Receptor Agonists

Synthesis and Structure–Activity Relationship Study of a New Series of Selective σ1 Receptor Ligands for the Treatment of Pain: 4-Aminotriazoles

Journal of Medicinal Chemistry ◽

10.1021/jm501920g ◽

2015 ◽

Vol 58 (5) ◽

pp. 2441-2451 ◽

Cited By ~ 27

Author(s):

José Luis Díaz ◽

Ute Christmann ◽

Ariadna Fernández ◽

Antoni Torrens ◽

Adriana Port ◽

...

Keyword(s):

Activity Relationship ◽

Receptor Ligands ◽

Σ1 Receptor ◽

Structure Activity ◽

Design and Synthesis of a Piperidinone Scaffold as an Analgesic through Kappa-Opioid Receptor: Structure–Activity Relationship Study of Matrine Alkaloids

Chemical and Pharmaceutical Bulletin ◽

10.1248/cpb.c15-00962 ◽

2016 ◽

Vol 64 (5) ◽

pp. 410-419 ◽

Cited By ~ 6

Author(s):

Hiroyoshi Teramoto ◽

Takayasu Yamauchi ◽

Yasushi Terado ◽

Sanae Odagiri ◽

Shigeru Sasaki ◽

...

Keyword(s):

Opioid Receptor ◽

Kappa Opioid Receptor ◽

Activity Relationship ◽

Kappa Opioid ◽

Design And Synthesis ◽

Receptor Structure ◽

Structure Activity ◽

Nascent structure–activity relationship study of a diastereomeric series of kappa opioid receptor antagonists derived from CJ-15,208

Bioorganic & Medicinal Chemistry Letters ◽

10.1016/j.bmcl.2009.04.105 ◽

2009 ◽

Vol 19 (13) ◽

pp. 3647-3650 ◽

Cited By ~ 24

Author(s):

Roland E. Dolle ◽

Mathieu Michaut ◽

Blanca Martinez-Teipel ◽

Pamela R. Seida ◽

Christopher W. Ajello ◽

...

Keyword(s):

Opioid Receptor ◽

Kappa Opioid Receptor ◽

Activity Relationship ◽

Receptor Antagonists ◽

Kappa Opioid ◽

Structure Activity ◽

Opioid Receptor Antagonists ◽

Structure–activity relationship study of a diverse set of estrogen receptor ligands (I) using MultiCASE expert system

Chemosphere ◽

10.1016/s0045-6535(02)00859-7 ◽

2003 ◽

Vol 51 (6) ◽

pp. 445-459 ◽

Cited By ~ 32

Author(s):

Gilles Klopman ◽

Suman K. Chakravarti

Keyword(s):

Estrogen Receptor ◽

Expert System ◽

Activity Relationship ◽

Receptor Ligands ◽

Structure Activity ◽

Relationship Study ◽

Estrogen Receptor Ligands

Structure activity relationship study of benzo[d]thiazol-2(3H)one based σ receptor ligands

Bioorganic & Medicinal Chemistry Letters ◽

10.1016/j.bmcl.2013.06.032 ◽

2013 ◽

Vol 23 (17) ◽

pp. 5011-5013 ◽

Cited By ~ 4

Author(s):

Rohit Bhat ◽

James A. Fishback ◽

Rae R. Matsumoto ◽

Jacques H. Poupaert ◽

Christopher R. McCurdy

Keyword(s):

Activity Relationship ◽

Receptor Ligands ◽

Structure Activity ◽

Development of κ Opioid Receptor Agonists by Focusing on Phenyl Substituents of 4-Dimethylamino-3-phenylpiperidine Derivatives: Structure–Activity Relationship Study of Matrine Type Alkaloids

Chemical and Pharmaceutical Bulletin ◽

10.1248/cpb.c15-00963 ◽

2016 ◽

Vol 64 (5) ◽

pp. 420-431 ◽

Cited By ~ 3

Author(s):

Hiroyoshi Teramoto ◽

Takayasu Yamauchi ◽

Shigeru Sasaki ◽

Kimio Higashiyama

Keyword(s):

Opioid Receptor ◽

Activity Relationship ◽

Receptor Agonists ◽

Structure Activity ◽

Relationship Study ◽

Opioid Receptor Agonists

Synthesis and Structure-Activity Relationship Study of 2-Substituted- 5-(5-nitro-2-thienyl)-1,3,4-thiadiazoles as Anti-Helicobacter pylori Agents

Letters in Drug Design & Discovery ◽

10.2174/157018009789057599 ◽

2009 ◽

Vol 6 (6) ◽

pp. 468-474 ◽

Cited By ~ 1

Author(s):

Alireza Foroumadi ◽

Somayeh Sedaghat ◽

Saeed Emami ◽

Maryam Yazdanian ◽

Mohammad Moshafi ◽

...

Keyword(s):

Helicobacter Pylori ◽

Activity Relationship ◽

Structure Activity ◽